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Compile Data Set for Download or QSAR
maximum 50k data
Found
13
Enz. Inhib. hit(s) with Target = 'Polycystin-1'
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86434
(12-Deoxyphorbol 13-phenylacetate | CAS_105100 | NS...)
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Affinity Data
Ki: 0.350nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86431
(CAS_4179 | Mezerein | NSC_4179)
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Affinity Data
Ki: 0.430nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86432
((-)-Octylindolactam V | CAS_159320 | NSC_159320)
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Affinity Data
Ki: 0.450nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86429
(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
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Affinity Data
Ki: 3.20nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86429
(CAS_6437389 | NSC_6437389 | Thymeleatoxin | Thymel...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.85nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86435
(B8-DL-B8 | B8-DL-B8 (low PS))
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Copy InChI
Affinity Data
Ki: 10.8nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86433
(CAS_454217 | NSC_454217 | Prostratin)
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Copy InChI
Affinity Data
Ki: 12.9nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86435
(B8-DL-B8 | B8-DL-B8 (low PS))
Copy SMILES
Copy InChI
Affinity Data
Ki: 26.1nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86430
((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
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Copy InChI
Affinity Data
Ki: 38nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86430
((-)-Indolactam V | (-)-Indolactam V (low PS) | CAS...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 48.1nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
PDB
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86436
(3-hydroxy-2-[4-methyl-3-(methylethyl)pentanoyloxy]...)
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Copy InChI
Affinity Data
Ki: 90nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM86440
(CAS_104731 | NSC_104731 | OAG)
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Copy InChI
Affinity Data
Ki: 146nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Polycystin-1
(Homo sapiens (Human))
University Of Pittsburgh
Curated by
PDSP K
i
Database
Ligand
BDBM50592745
(CHEMBL5188373)
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Affinity Data
IC50: 81nM
Assay Description:
Inhibition of PKD1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
PubMed
Copy BDB DOI